Shan Li,Tao Zhang,Su-Jie Zhu,Chong Lei,Mengzhen Lai,Lijie Peng,Linjiang Tong,Zilu Pang,Xiaoyun Lu,Jian Ding,Xiaomei Ren,Cai-Hong Yun,Hua Xie,Ke Ding,Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR(T790M/C797S) Mutants.ACS Med Chem Lett. 13(2):196-202 (2022).
https://doi.org/10.1021/acsmedchemlett.1c00555.